Inhibitor

Fondaparinux Sodium

Fondaprinux is sulfated pentasaccharide, an ultra low molecular weight synthetic form of heparain with antithrombotic properties.  It is analogous to the pentasaccharide sequence in heparin. Mechanism of Action Fondaprinux Sodium binds...

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Fumitremorgin B

  Molecular Formula  C27H33N3O5  

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Kazusamycin A

Kazusamycin A is a minor member of the Leptomycin complex isolated from some Streptomyces species. It is a hydroxylated analog of Leptomycin B, a nuclear export inhibitor. It is similar to Leptomycins A and B in physico-chemical and biological...

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Kazusamycin B

Kazusamycin B is a metabolite and minor member of the Leptomycin complex isolated from some Streptomyces species. It is a hydroxylated analog of Leptomycin A, a nuclear export inhibitor. It is similar to Leptomycins A and B in physico-chemical and...

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Leptomycin B

Leptomycin B is the dominant member of the Leptomycin class, secondary metabolites isolated from selected Streptomyces strains.  It is a bioactive small molecule with antifungal and antibacterial activity.  It is a nuclear export inhibitor,...

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Levodropropizine

Levodropropizine has anti-allergic properties and inhibits the histamine receptor. It acts as a peripheral antitussive agent. Mechanism of Action Levodropropizine has affinity for H1-histaminic and alpha-adrenergic receptors. Levodropropizine has a...

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Levofloxacin Hydrochloride

Levofloxacin HCl is the hydrochloride salt of Levofloxacin.  It is a broad-spectrum fluoroquinolone antibiotic and the optical S-(-) isomer of Ofloxacin. The compound is a DNA gyrase inhibitor, and has been shown to inhibit topoisomerase IV. ...

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Meropenem Vaborbactam (1:1 mixture)

Meropenem Vaborbactam (1:1 mixture) is a mixture of Meropenem (a carbapenem antibiotic) and Vaborbactam (a cyclic, boronic acid-based, non-suicidal, reversible beta-lactamase inhibitor). It is active against the bacteria causing complicated urinary tract...

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Methylspinazarin

Methylspinazarin is a rare naphthoquinone pigment produced by a strain of Streptomyces filipinensis, isolated by Nagatsu and colleagues at Ochanomizu University, Japan in 1973. Methylspinazarin inhibits catechol-O-methyl transferase (COMT) and exhibits a...

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Miconazole Nitrate

Miconazole Nitrate is the nitrate salt of Miconazole, an imidazole antimycotic compound patented in 1968 (Janssen Pharmaceutica).  It targets the fungi that cause tinea (ringworm) and athlete’s foot.  It inhibits ergosterol synthesis, and...

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Monomethylsulochrin

Monomethylsulochrin is a benzophenone isolated from Aspergillus fumigatus by Turner, ICI Ltd in 1965. Monomethylsulochrin inhibits eosinophil degranulation. Its dimethyl analogue, sulochrin, inhibits VEGF leading to inhibition of capillary-like tube...

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Multiflorenol

Multiflorenol is a triterpenoid found in the geranium family and other flowering plants, first isolated and the structure elucidated by Khastgir and Sengupta in 1961. Multiflorenol was subsequently isolated by Ritchie and Taylor from the Australian...

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